Cabergoline: All You Need When Bodybuilding
In this instance, a Cabergoline oral tablet is a prescription medication that is only available as a generic medication. There is currently no brand-name version of this product available. Cabergoline is only available as a tablet that must be swallowed.
What it is used for
Cabergoline is a medication that is used to treat hyperprolactinemia (high levels of prolactin in your body). This occurs when your pituitary gland produces an excessive amount of prolactin. A problem with your hormones or a tumor in your pituitary gland could be the cause of your elevated prolactin levels.
Ovulation, the menstrual cycle, and the production of breast milk can all be affected by high prolactin levels in a woman’s body. Prolactin levels that are too high in men can interfere with reproduction and cause sexual problems. These difficulties include a decreased sex drive as well as the inability to obtain or maintain an erection.
The pituitary gland is responsible for the production of prolactin. It aids in the stimulation and maintenance of breast milk production. Hyperprolactinemia is a condition in which a person’s body produces an excessive amount of this hormone.
The presence of this ailment during pregnancy or while producing milk for nursing is considered normal.
Hyperprolactinemia, on the other hand, may occur in anybody due to certain medical conditions or the use of particular drugs. The causes and consequences of elevated prolactin levels differ depending on the gender of the individual.
It is possible that an elevated level of prolactin is produced by a number of secondary diseases. The majority of the time, hyperprolactinemia is caused by pregnancy, which is completely natural.
In a 2013 research, it was shown that pituitary tumors may be responsible for roughly 50 percent of all cases of hyperprolactinemia. A prolactinoma is a tumor that develops in the pituitary gland, which produces the hormone prolactin. These tumors are almost often noncancerous in nature. However, they may create symptoms that vary depending on the gender of the individual who is experiencing them.
Other factors that contribute to hyperprolactinemia include:
- Acid H2 blockers, such as cimetidine (Tagamet)
- Antihypertensive medications, such as verapamil (Calan, Isoptin, and Verelan)
- Cirrhosis, or severe scarring of the liver
- Cushing syndrome, which can result from high levels of the hormone cortisol
- Infection, tumor, or trauma of the hypothalamus
- Anti-nausea medication such as metoclopramide (Primperan, Reglan)
- Antidepressant drugs such as desipramine (Norpramin) and clomipramine
Hyperprolactinemia is characterized by the presence of certain symptoms.
Men and women may have different signs and symptoms of hyperprolactinemia.
Because prolactin levels impact both milk production and menstrual periods, it might be difficult to identify in males with low prolactin levels. If a guy is suffering from erectile dysfunction, his doctor may prescribe that he have a blood test to check for an excess of the hormone prolactin.
Symptoms experienced by females include:
- Periods that are erratic
- Alterations in menstrual flow
- A break in the menstrual cycle
- Lactation causes a decrease in libido (galactorrhea)
- A burning sensation in the breasts
- A feeling of dryness in the vaginal area
Symptoms in men include:
- Atypical breast development (gynecomastia)
- A decrease in sexual desire
- Vision problems
What is the procedure for diagnosing hyperprolactinemia?
A blood test to assess prolactin levels is performed by a doctor in order to identify hyperprolactinemia.
If prolactin levels are high, the doctor will order more tests to rule out other diseases. Whether they have reason to believe a tumor is there, they may request an MRI scan to see if a pituitary tumor is really present.
Diagnosis and management of hyperprolactinemia
The majority of hyperprolactinemia treatments are geared around restoring prolactin levels to normal levels. Even though surgery may be required to remove a prolactinoma tumor in certain cases, the illness is generally treatable with medication.
The following procedures may be used in treatment:
- Change of medication
- Synthetic thyroid hormones
- Medication to reduce prolactin, such as bromocriptine (Parlodel, Cycloset) or cabergoline
See also Letrozole: Main Benefits, Proper Dosage, Cycle and Risks
How does it work?
Cabergoline is a drug that belongs to a class of medications known as dopamine agonists. A class of drugs is a collection of medications that have similar mechanisms of action. These medications are frequently used to treat conditions that are very similar to one another.
Dopamine is a chemical produced by your body. It works by preventing your body from producing prolactin. Cabergoline works by attaching itself to dopamine receptors in the brain. This also prevents your body from releasing prolactin, which aids in the reduction of your prolactin levels in the blood.
It is generated predominantly by the pituitary gland, which is responsible for its function. Prolactin, also known as lactotropin, is a hormone that allows animals, particularly females, to create milk by stimulating the production of milk. As well as impacting behavior and regulating the immune system, prolactin is involved in a variety of other physiological activities, including those related to breastfeeding.
Excess prolactin in males might cause symptoms such as the following:
- Breasts that have grown in size
- Nipple discharge
- Erectile dysfunction
- sex desire at a low level
- a reduction in the amount of body hair
- Low testosterone levels are a problem
Hyperprolactinemia is a medical term that refers to elevated amounts of prolactin in the blood. High levels of prolactin in women may result in symptoms such as irregular periods, excessive breast milk, infertility, and breast discomfort, among other things.
Is Cabergoline beneficial to one’s sexual health?
Cabergoline is a drug that has the potential to be beneficial in helping men control the symptoms of excessive prolactin levels. The following are some of its advantages for sexual health:
Male Orgasmic Disorder (MOD): What to expect and how to treat It
Male orgasmic dysfunction is defined as the lack of orgasm during sexual encounters on a consistent or regular basis. Male orgasmic dysfunction may be caused by a variety of medical disorders, the most common of which is elevated prolactin levels.
Researchers believe cabergoline may be an effective therapy for male orgasmic problems and delayed orgasm, independent of the patient’s age or the source of his illness.
A Medication for Erectile Dysfunction that is used in conjunction with other medications
Erectile Dysfunction (ED) is characterized by the inability to get or sustain a firm erection as a result of a combination of physiological and psychological causes. ED itself, as well as its underlying physiological or psychogenic causes, may result in unpleasant sex life, poor self-esteem, marital issues, stress, and anxiety in the sufferer and those around him.
When used in conjunction with tadalafil medication, cabergoline has been demonstrated to be a safer and more effective therapy option for individuals with psychogenic erectile dysfunction when compared to treatment with tadalafil alone.
It may be possible to raise testosterone levels using this supplement.
Because of variables such as an increase in comorbidities or current diseases, as well as the aging population, testosterone levels in men normally decline over time.
Reduced sex desire, sadness, poor mental performance, lack of energy, erectile dysfunction, and osteoporosis are all connected with testosterone shortage in older men, as is the loss of muscle mass and strength.
Prolactin levels that are too high in males cause testosterone levels to drop.
According to research, long-term therapy with cabergoline has been demonstrated to lower prolactin levels while simultaneously increasing testosterone levels by a substantial amount. Aside from that, following six months of therapy, sperm health has increased in terms of volume and quantity as well as quick advancement and motility.
Side effects of Cabergoline
It is possible to experience nausea, vomiting, stomach upset, constipation, dizziness, lightheadedness, or fatigue. Inform your doctor or pharmacist as soon as possible if any of these side effects persist or worsen.
Please keep in mind that this medication has been prescribed by your doctor because he or she has determined that the benefit to you outweighs the risk of side effects. The majority of people who take this medication do not experience any serious side effects.
In the event that any of the following rare but serious side effects occur: persistent cough, mental/emotional changes (such as nervousness), unusually strong urges (such as increased gambling, increased sexual urges), vision changes, painful menstrual periods, breast pain, symptoms of heart failure (such as shortness of breath, swelling ankles/feet, unusual tiredness, unusual/sudden weight gain), contact your doctor immediately.
If you experience any serious side effects, such as chest pain or signs of kidney problems (such as a change in the amount of urine produced or lower back/flanking pain), seek medical attention right away.
It is extremely rare for this medication to cause a life-threatening allergic reaction. However, seek immediate medical attention if you experience any of the following symptoms of a serious allergic reaction: rash, itching/swelling (especially of the face, tongue, or throat), severe dizziness, or difficulty breathing.
Precautions Before taking Cabergoline
You should tell your doctor or pharmacist if you are allergic to cabergoline, if you are allergic to other ergot medications (such as ergotamine), or if you have any other allergies before taking this medication. It is possible that this product contains inactive chemicals that might cause allergic reactions or other complications. For more information, consult with your pharmacist.
If you have a medical history that includes liver disease, high blood pressure (hypertension), heart valve disease, abnormal scarring or thickening of the lining of the lungs, heart, or abdomen (pulmonary/pericardial/retroperitoneal fibrosis), tell your doctor or pharmacist before using this medication.
This medication may cause you to feel dizzy. You may become dizzier if you consume alcohol or marijuana (cannabis). Do not drive, operate equipment, or engage in any activity that requires attentiveness until you are certain that you can do so safely. Keep alcoholic drinks to a minimum. If you are a marijuana user, you should consult with your doctor (cannabis).
When getting out of a sitting or lying position, get up slowly to reduce the likelihood of experiencing dizziness or lightheadedness.
Before having surgery, inform your doctor or dentist of all of the products you use on a daily basis (including prescription drugs, nonprescription drugs, and herbal products).
See also The Exemestane Guide: How It Works, Positive Effects, and Warnings
Cabergoline dosage and administration
Before you begin treatment, make sure you have read the written information sheet provided by the manufacturer, which may be found within the package. It will offer you further information on cabergoline as well as a comprehensive list of the negative effects that you may encounter as a result of taking it.
The amount of cabergoline you will need to take will be determined by the reason you are taking it. If you are using cabergoline to decrease high prolactin levels, you may only need one dosage each week if you are just taking it for a few days to end breast milk. If you have Parkinson’s disease, you may only need one dose per day if you are taking cabergoline to lower high prolactin levels. To help you remember how much and how frequently to take it, your doctor will tell you how much and how often to take it. This information will also be put on the label of the package to remind you.
Read your doctor’s instructions carefully and take cabergoline precisely as he or she instructs you to. For the first time, your doctor may prescribe a tiny dosage of cabergoline and then gradually raise the amount you take each day. Gradually raising your dosage in this manner can help to prevent the occurrence of adverse effects such as dizziness, which may occur during the initial few days of therapy.
Take the pill with a glass of water at the beginning of a meal. It is recommended to take cabergoline after a meal to lessen the likelihood of feeling unwell (nausea).
When taking cabergoline, try to take it at the same time(s) each day; if you are taking it on a weekly basis, try to take it on the same day (or days) each week.
You should take your medication as soon as you remember if you forget to take it. If you realize that you missed dosage and it is almost time for your next dose, take your next dose when it is due but skip the dose that you missed. Do not take two doses at the same time to make up for a missed dosage.
The advantages of using Cabergoline in bodybuilding
Even some of the most seasoned bodybuilders in the world, who have been utilizing SARMs (Selective Androgen Receptor Modulators) for years, had never heard of cabergoline until recently. So what I would want to do here is speak to you about the advantages and disadvantages of utilizing cabergoline for bodybuilding, as well as the risks involved.
Many of the cabergoline reviews that are available online are very positive. Now, just like every other review out there, I will tell you that it is all you need both as a PCT supplement (often a Selective Estrogen Receptor Modulator) and as a dopamine-stimulating motivating tablet and that it is the best of both worlds.
How Cabergoline is beneficial for bodybuilding
It acts by inhibiting the generation of prolactin in the female reproductive system. Prolactin plays an important role in a variety of functions in the body, particularly in the female body. In general, lowering the company’s output has a number of advantages.
Because it reduces the synthesis of prolactin, it aids in the suppression of the most severe adverse effects of testosterone-stimulating medications such as SARMs, making it an excellent PCT supplement in conjunction with Nolvadex or Clomid (both Selective Estrogen Receptor Modulators).
In contrast to Nolvadex or Clomid, cabergoline is not a synthetic estrogenic receptive modulator (SERM). As a result of taking cabergoline, the pituitary gland is instructed to produce less prolactin, which results in a reduction in milk production. Dopamine production is increased as a result of this.
Dopamine is essential to our ability to perform in the gym since it is our primary reward and dangerous hormone. When it is released, you should push yourself harder to attain your objectives and feel better when you do so.
In addition, since cabergoline reduces the synthesis of prolactin, it enables a higher amount of testosterone to be produced. Along with this, there is the fact that increased dopamine production results in more physical aggressiveness, which translates into tougher exercises and performance, which in turn results in increased testosterone production.
The effects and advantages of Cabergoline in the bodybuilding industry
Taking everything into consideration, the following are the favorable effects of utilizing cabergoline for bodybuilding:
Because of the increased amounts of dopamine production, you will be more motivated and more concentrated in your efforts to attain your bodybuilding objectives, both during individual exercises and over the long term. After a few days, you will surely notice a surge in dopamine levels. You will be able to push yourself harder as time goes on, and you will feel very driven as a result.
Because of the increased levels of dopamine production, as well as the decreased levels of prolactin, you will be able to sustain greater testosterone levels even when the SARMs you are taking are suppressing them.
Cabergoline may be used as a PCT supplement in conjunction with other drugs.
It can be used alone or in combination with Nolvadex or Clomid to increase motivation and upbeat feelings, which can help to offset the negative effects of low testosterone levels. It also works to increase testosterone production by inhibiting the release of prolactin, which helps to raise testosterone levels.
Overall, cabergoline has the potential to be beneficial to bodybuilders both throughout their cycle and as part of their post-cycle treatment. It has worked well for me over the last couple of years; however, I do take it in moderation and recommend that you do as well.
Cabergoline dosage(for bodybuilding) and half-Life
For the record, one thing I would want to make clear to you is that there is no fixed range of cabergoline dosages for you to work within since as you are now aware, cabergoline was not intended for bodybuilding usage in the first place.
However, it is a very strong substance. Sometimes it is recommended in quantities of roughly 50 mcg, which is micrograms rather than milligrams, so you must be very cautious while administering the medication.
Also, keep in mind that the half-life of cabergoline is rather lengthy, around three days, which is much longer than the half-life of most other supplements on the market. That means you just need to administer this medication a couple of times each week to gain the advantages of increased dopamine and testosterone levels.
It is available from Swiss Chems, where it is dosed at 50 mcg each pill, which is pretty much optimal in my opinion.
However, I would caution that it is not a good PCT supplement to use on its own, since it is not recommended. You will see a rise in your testosterone levels, as well as an increase in your dopamine levels.
Nonetheless, it is critical for me to inform you that its capacity to lower estrogen levels is not as effective as that of Nolvadex or Clomid. As a result, running it on its own during PCT is not recommended.
My recommendation is to take 50 mcg twice a week in addition to your regular Nolvadex dosage. As a result, you will experience a big increase in testosterone and dopamine, as well as a considerable decrease in estrogen levels. For the greatest overall post-cycle therapeutic results, you will need to stack it with a modest dosage of Nolvadex or Clomid, which means you will need to stack it with both.
A large number of men utilize it while riding their bicycles. I honestly would not stack it with SARMs at the same dosage you would take it between cycles, while it is possible.
On cycle, I would recommend that you run it at the lower 25 mcg dosage twice per week rather than three times per week. The dopamine and testosterone enhancing effects of this method will help you become more aggressive and determined, while also helping to maintain your testosterone levels high towards the end of your cycle and not imbalance you too much for the rest of your cycle.
See also Anastrozole: How This Breast Cancer Drug Can Slow Progression of the Disease